Ligand source activities (1 row/activity)
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
|
| 10883396 | 3649 | None | 30 | Human | Functional | pEC50 | = | 6.1 | 6.1 | -562 | 15 | Guide to Pharmacology | 379 | 17 | 4 | 4 | 4.0 | CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O | 12618218 | |||
| 5283560 | 3649 | None | 30 | Human | Functional | pEC50 | = | 6.1 | 6.1 | -562 | 15 | Guide to Pharmacology | 379 | 17 | 4 | 4 | 4.0 | CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O | 12618218 | |||
| 911 | 3649 | None | 30 | Human | Functional | pEC50 | = | 6.1 | 6.1 | -562 | 15 | Guide to Pharmacology | 379 | 17 | 4 | 4 | 4.0 | CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O | 12618218 | |||
| CHEMBL225155 | 3649 | None | 30 | Human | Functional | pEC50 | = | 6.1 | 6.1 | -562 | 15 | Guide to Pharmacology | 379 | 17 | 4 | 4 | 4.0 | CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O | 12618218 | |||
| 2921 | 1422 | None | 0 | Human | Functional | pEC50 | = | 6.2 | 6.2 | -67 | 2 | Guide to Pharmacology | 381 | 18 | 4 | 4 | 4.3 | CCCCCCCCCCCCCCC[C@H]([C@H](COP(=O)(O)O)N)O | 12618218 | |||
| 44317142 | 1422 | None | 0 | Human | Functional | pEC50 | = | 6.2 | 6.2 | -67 | 2 | Guide to Pharmacology | 381 | 18 | 4 | 4 | 4.3 | CCCCCCCCCCCCCCC[C@H]([C@H](COP(=O)(O)O)N)O | 12618218 | |||
| 644260 | 1422 | None | 0 | Human | Functional | pEC50 | = | 6.2 | 6.2 | -67 | 2 | Guide to Pharmacology | 381 | 18 | 4 | 4 | 4.3 | CCCCCCCCCCCCCCC[C@H]([C@H](COP(=O)(O)O)N)O | 12618218 | |||
| CHEMBL78494 | 1422 | None | 0 | Human | Functional | pEC50 | = | 6.2 | 6.2 | -67 | 2 | Guide to Pharmacology | 381 | 18 | 4 | 4 | 4.3 | CCCCCCCCCCCCCCC[C@H]([C@H](COP(=O)(O)O)N)O | 12618218 | |||
| 5512 | 1430 | None | 0 | Human | Functional | pEC50 | = | 6.3 | 6.3 | - | 1 | Guide to Pharmacology | 701 | 36 | 2 | 6 | 11.6 | CCCCCCCC/C=C\CCCCCCCC(=O)OCC(OC(=O)CCCCCCC/C=C\CCCCCCCC)COP(=O)(O)O | 12618218 | |||
| 9547172 | 1430 | None | 0 | Human | Functional | pEC50 | = | 6.3 | 6.3 | - | 1 | Guide to Pharmacology | 701 | 36 | 2 | 6 | 11.6 | CCCCCCCC/C=C\CCCCCCCC(=O)OCC(OC(=O)CCCCCCC/C=C\CCCCCCCC)COP(=O)(O)O | 12618218 | |||
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
|